2924546-70-1
2924546-70-1 structure
- Name: SJ1461
- Chemical Name: SJ1461
- CAS Number: 2924546-70-1
- Molecular Formula: C21H18ClN7OS2
- Molecular Weight: 484.00
- Catalog: Signaling Pathways Epigenetics Epigenetic Reader Domain
- Create Date: 2023-09-19 11:19:10
- Modify Date: 2024-01-02 19:44:30
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SJ1461 is a potent and orally active BET inhibitor. SJ1461 inhibits BRD2 (BD1), and BRD2 (BD2), BRD4 (BD1), and BRD4 (BD2) with IC50 values of 1.6 nM, 0.1 nM, 6.5 nM, and 0.2 nM, respectively[1].
| Name | SJ1461 |
|---|
| Description | SJ1461 is a potent and orally active BET inhibitor. SJ1461 inhibits BRD2 (BD1), and BRD2 (BD2), BRD4 (BD1), and BRD4 (BD2) with IC50 values of 1.6 nM, 0.1 nM, 6.5 nM, and 0.2 nM, respectively[1]. |
|---|---|
| Related Catalog | |
| Target |
BRD2 (BD1):1.6 nM (IC50) BRD2 (BD2):0.1 nM (IC50) BRD4 (BD1):6.5 nM (IC50) BRD4 (BD2):0.2 nM (IC50) |
| References |
| Molecular Formula | C21H18ClN7OS2 |
|---|---|
| Molecular Weight | 484.00 |