![]() GSK217 structure
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Common Name | GSK217 | ||
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CAS Number | 2748687-92-3 | Molecular Weight | 360.421 | |
Density | N/A | Boiling Point | N/A | |
Molecular Formula | C20H20N6O | Melting Point | N/A | |
MSDS | N/A | Flash Point | N/A |
Use of GSK217GSK217 (GSK-217) is a potent, highly selective BET BD2 inhibitor with pIC50 of 7.5 (BRD4 BD2), 300-fold selectivity over BRD4 BD1. |
Name | GSK217 |
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Description | GSK217 (GSK-217) is a potent, highly selective BET BD2 inhibitor with pIC50 of 7.5 (BRD4 BD2), 300-fold selectivity over BRD4 BD1. |
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References | 1. Helen E Aylott, et al. J Med Chem. 2021 Mar 25;64(6):3249-3281. |
Molecular Formula | C20H20N6O |
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Molecular Weight | 360.421 |