GSK217

Modify Date: 2024-04-09 11:59:35

GSK217 Structure
GSK217 structure
Common Name GSK217
CAS Number 2748687-92-3 Molecular Weight 360.421
Density N/A Boiling Point N/A
Molecular Formula C20H20N6O Melting Point N/A
MSDS N/A Flash Point N/A

 Use of GSK217


GSK217 (GSK-217) is a potent, highly selective BET BD2 inhibitor with pIC50 of 7.5 (BRD4 BD2), 300-fold selectivity over BRD4 BD1.

 Names

Name GSK217

 GSK217 Biological Activity

Description GSK217 (GSK-217) is a potent, highly selective BET BD2 inhibitor with pIC50 of 7.5 (BRD4 BD2), 300-fold selectivity over BRD4 BD1.
References 1. Helen E Aylott, et al. J Med Chem. 2021 Mar 25;64(6):3249-3281.

 Chemical & Physical Properties

Molecular Formula C20H20N6O
Molecular Weight 360.421
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