GSK217

Names

[ Name ]:
GSK217

Biological Activity

[Description]:

GSK217 (GSK-217) is a potent, highly selective BET BD2 inhibitor with pIC50 of 7.5 (BRD4 BD2), 300-fold selectivity over BRD4 BD1.

[References]

1. Helen E Aylott, et al. J Med Chem. 2021 Mar 25;64(6):3249-3281.

Chemical & Physical Properties

[ Molecular Formula ]:
C₂₀H₂₀N₆O

[ Molecular Weight ]:
360.421

Related Compounds

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