2748687-92-3
2748687-92-3 structure
- Name: GSK217
- Chemical Name: GSK217
- CAS Number: 2748687-92-3
- Molecular Formula: C20H20N6O
- Molecular Weight: 360.421
- Catalog: Signaling Pathways Epigenetics Epigenetic Reader Domain
- Create Date: 2022-07-02 13:07:50
- Modify Date: 2024-04-09 11:59:35
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GSK217 (GSK-217) is a potent, highly selective BET BD2 inhibitor with pIC50 of 7.5 (BRD4 BD2), 300-fold selectivity over BRD4 BD1.
| Name | GSK217 |
|---|
| Description | GSK217 (GSK-217) is a potent, highly selective BET BD2 inhibitor with pIC50 of 7.5 (BRD4 BD2), 300-fold selectivity over BRD4 BD1. |
|---|---|
| References | 1. Helen E Aylott, et al. J Med Chem. 2021 Mar 25;64(6):3249-3281. |
| Molecular Formula | C20H20N6O |
|---|---|
| Molecular Weight | 360.421 |