Tabimorelin hemifumarate

Modify Date: 2024-02-25 13:45:42

Tabimorelin hemifumarate structure	Common Name	Tabimorelin hemifumarate
	CAS Number	242143-80-2	Molecular Weight	586.72
	Density	N/A	Boiling Point	N/A
	Molecular Formula	C₃₂H₄₀N₄O_3.1/₂C₄H₄O₄	Melting Point	N/A
	MSDS	N/A	Flash Point	N/A

Use of Tabimorelin hemifumarate

Tabimorelin (NN703) hemifumarate is an orally active growth hormone (GH) secretagogue. Tabimorelin hemifumarate is also a potent inhibitor of CYP3A4 activity[1].

Name	Tabimorelin hemifumarate
Synonym	More Synonyms

Description	Tabimorelin (NN703) hemifumarate is an orally active growth hormone (GH) secretagogue. Tabimorelin hemifumarate is also a potent inhibitor of CYP3A4 activity[1].
Related Catalog	Research Areas >> Endocrinology Signaling Pathways >> Metabolic Enzyme/Protease >> Cytochrome P450
Target	CYP3A4
References	[1]. Zdravkovic M, et al. A clinical study investigating the pharmacokinetic interaction between NN703 (tabimorelin), a potential inhibitor of CYP3A4 activity, and midazolam, a CYP3A4 substrate. Eur J Clin Pharmacol. 2003 Feb;58(10):683-8.

Molecular Formula	C₃₂H₄₀N₄O_3.1/₂C₄H₄O₄
Molecular Weight	586.72
Exact Mass	1172.630981

D-Phenylalaninamide, N-[(2E)-5-amino-5-methyl-1-oxo-2-hexen-1-yl]-N-methyl-3-(2-naphthalenyl)-D-alanyl-N,Nα-dimethyl-, (2E)-2-butenedioate (2:1)

N-[(2E)-5-Amino-5-methyl-2-hexenoyl]-N-methyl-3-(2-naphthyl)-D-alanyl-N,Nα-dimethyl-D-phenylalaninamide (2E)-2-butenedioate (2:1)

Tabimorelin

N-[(2E)-5-Amino-5-methylhex-2-enoyl]-N-methyl-3-(2-naphthyl)-D-alanyl-N,Nα-dimethyl-D-phenylalaninamide (2E)-but-2-enedioate (2:1)

Tabimorelin hemifumarate

Use of Tabimorelin hemifumarate

Names

Tabimorelin hemifumarate Biological Activity

Chemical & Physical Properties

Synonyms