P2Y2R/GPR17 antagonist 1

Modify Date: 2025-09-13 18:25:32

P2Y2R/GPR17 antagonist 1 Structure
P2Y2R/GPR17 antagonist 1 structure
 Common Name P2Y2R/GPR17 antagonist 1
CAS Number 2395016-49-4 Molecular Weight 432.83
Density N/A Boiling Point N/A
Molecular Formula C19H13ClN2O6S Melting Point N/A
MSDS N/A Flash Point N/A

 Use of P2Y2R/GPR17 antagonist 1


P2Y2R/GPR17 antagonist 1 (Compound 14m) is a dual P2Y2R and GPR17 antagonist with IC50 values of 3.17 µM and 1.67 µM against P2Y2R and GPR17, respectively. P2Y2R/GPR17 antagonist 1 shows excellent metabolic stability in human liver microsomes[1].

 Names

Name P2Y2R/GPR17 antagonist 1

 P2Y2R/GPR17 antagonist 1 Biological Activity

Description P2Y2R/GPR17 antagonist 1 (Compound 14m) is a dual P2Y2R and GPR17 antagonist with IC50 values of 3.17 µM and 1.67 µM against P2Y2R and GPR17, respectively. P2Y2R/GPR17 antagonist 1 shows excellent metabolic stability in human liver microsomes[1].
Related Catalog
Target

IC50: 1.67 µM (GPR17), 3.17 µM (P2Y2R)[1]

References

[1]. Pillaiyar T, et al. Design, synthesis and biological evaluation of suramin-derived dual antagonists of the proinflammatory G protein-coupled receptors P2Y2 and GPR17. Eur J Med Chem. 2020 Jan 15;186:111789.

 Chemical & Physical Properties

Molecular Formula C19H13ClN2O6S
Molecular Weight 432.83
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