RTICBM-229

Modify Date: 2024-08-13 14:38:59

RTICBM-229 Structure
RTICBM-229 structure
Common Name RTICBM-229
CAS Number 2250355-35-0 Molecular Weight 311.769
Density N/A Boiling Point N/A
Molecular Formula C17H14ClN3O Melting Point N/A
MSDS N/A Flash Point N/A

 Use of RTICBM-229


RTICBM-229 is a potent, selective, brain-penetrant CB1 negative allosteric modulator (NAM) with IC50 of 169 nM in Ca2+ assay, 40 nM in GTPγS assay.

 Names

Name RTICBM-229

 RTICBM-229 Biological Activity

Description RTICBM-229 is a potent, selective, brain-penetrant CB1 negative allosteric modulator (NAM) with IC50 of 169 nM in Ca2+ assay, 40 nM in GTPγS assay.
References 1. Thuy Nguyen, et al. J Med Chem. 2019 Nov 14;62(21):9806-9823.

 Chemical & Physical Properties

Molecular Formula C17H14ClN3O
Molecular Weight 311.769
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