Deltasonamide 1 TFA structure
|
Common Name | Deltasonamide 1 TFA | ||
|---|---|---|---|---|
| CAS Number | 2235358-73-1 | Molecular Weight | 761.27 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C32H40ClF3N6O6S2 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of Deltasonamide 1 TFADeltasonamide 1 TFA is a PDE6δ-KRas inhibitor. Deltasonamide 1 can inhibit PDE6δ-KRas with a KD of 203 pM. Deltasonamide 1 can be used for the research of tumors[1]. |
| Name | Deltasonamide 1 TFA |
|---|
| Description | Deltasonamide 1 TFA is a PDE6δ-KRas inhibitor. Deltasonamide 1 can inhibit PDE6δ-KRas with a KD of 203 pM. Deltasonamide 1 can be used for the research of tumors[1]. |
|---|---|
| Related Catalog | |
| Target |
KD: 203 pM (PDE6δ-KRas)[1] |
| In Vitro | Deltasonamide 1 可以抑制 PDE6δ-KRas,KD 为 203 pM[1]。 Deltasonamide 1 通过多达 7 个氢键与 PDE6δ 结合,产生皮摩尔亲和力[1]。 Deltasonamide 1 强烈减少增殖[1]。 Cell Proliferation Assay[1] Cell Line: RTCA of hPDAC cell lines Concentration: 0.375, 0.75, 1.5, 3, 6, 12 μM Incubation Time: 60 h Result: Inhibited proliferation of human pancreatic cancer cell lines. |
| References |
| Molecular Formula | C32H40ClF3N6O6S2 |
|---|---|
| Molecular Weight | 761.27 |