Deltasonamide 1 TFA

Modify Date: 2024-04-02 19:40:13

Deltasonamide 1 TFA Structure
Deltasonamide 1 TFA structure
 Common Name Deltasonamide 1 TFA
CAS Number 2235358-73-1 Molecular Weight 761.27
Density N/A Boiling Point N/A
Molecular Formula C32H40ClF3N6O6S2 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of Deltasonamide 1 TFA


Deltasonamide 1 TFA is a PDE6δ-KRas inhibitor. Deltasonamide 1 can inhibit PDE6δ-KRas with a KD of 203 pM. Deltasonamide 1 can be used for the research of tumors[1].

 Names

Name Deltasonamide 1 TFA

 Deltasonamide 1 TFA Biological Activity

Description Deltasonamide 1 TFA is a PDE6δ-KRas inhibitor. Deltasonamide 1 can inhibit PDE6δ-KRas with a KD of 203 pM. Deltasonamide 1 can be used for the research of tumors[1].
Related Catalog
Target

KD: 203 pM (PDE6δ-KRas)[1]

In Vitro Deltasonamide 1 可以抑制 PDE6δ-KRas，KD 为 203 pM[1]。 Deltasonamide 1 通过多达 7 个氢键与 PDE6δ 结合，产生皮摩尔亲和力[1]。 Deltasonamide 1 强烈减少增殖[1]。 Cell Proliferation Assay[1] Cell Line: RTCA of hPDAC cell lines Concentration: 0.375, 0.75, 1.5, 3, 6, 12 μM Incubation Time: 60 h Result: Inhibited proliferation of human pancreatic cancer cell lines.
References

[1]. Pablo Martín-Gago, et al. A PDE6δ-KRas Inhibitor Chemotype With Up to Seven H-Bonds and Picomolar Affinity That Prevents Efficient Inhibitor Release by Arl2. Angew Chem Int Ed Engl. 2017 Feb 20;56(9):2423-2428.  

 Chemical & Physical Properties

Molecular Formula C32H40ClF3N6O6S2
Molecular Weight 761.27
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