β2AR/M-receptor agonist-1
Modify Date: 2024-01-12 17:24:04
β2AR/M-receptor agonist-1 structure
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Common Name | β2AR/M-receptor agonist-1 | ||
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| CAS Number | 2230520-62-2 | Molecular Weight | 806.82 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C43H56BrN3O7 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of β2AR/M-receptor agonist-1β2AR/M-receptor agonist-1 (example 131) is a muscarinic antagonist and β2 adrenoceptor agonist (MABA). β2AR/M-receptor agonist-1 shows potency to β2 adrenoceptor with an EC50 value of 9.2 nM. β2AR/M-receptor agonist-1 also has potency to muscarinic receptor with a Ki value of 30.2 nM. β2AR/M-receptor agonist-1 shows MABA potency with an EC50 value of 4.0 nM[1]. |
| Name | β2AR/M-receptor agonist-1 |
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| Description | β2AR/M-receptor agonist-1 (example 131) is a muscarinic antagonist and β2 adrenoceptor agonist (MABA). β2AR/M-receptor agonist-1 shows potency to β2 adrenoceptor with an EC50 value of 9.2 nM. β2AR/M-receptor agonist-1 also has potency to muscarinic receptor with a Ki value of 30.2 nM. β2AR/M-receptor agonist-1 shows MABA potency with an EC50 value of 4.0 nM[1]. |
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| Related Catalog | |
| In Vivo | β2AR/M-receptor agonist-1 (0.01 和 0.1 mg/kg；静脉注射，一次) 降低比格犬的心率[1]。 |
| References |
| Molecular Formula | C43H56BrN3O7 |
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| Molecular Weight | 806.82 |