β2AR/M-receptor agonist-2

Modify Date: 2025-08-25 13:32:37

β2AR/M-receptor agonist-2 structure	Common Name	β2AR/M-receptor agonist-2
	CAS Number	1017857-38-3	Molecular Weight	717.31
	Density	N/A	Boiling Point	N/A
	Molecular Formula	C₃₆H₄₉ClN₄O₇S	Melting Point	N/A
	MSDS	N/A	Flash Point	N/A

Use of β2AR/M-receptor agonist-2

β2AR/M-receptor agonist-2 (compound 15) is a muscarinic antagonist and β2 adrenoceptor agonist (MABA). β2AR/M-receptor agonist-2 shows potency to β2 adrenoceptor with an EC50 value of 3.7 nM. β2AR/M-receptor agonist-2 also has potency to human cloned M3 receptor with a Ki value of 0.73 nM. β2AR/M-receptor agonist-2 is a potent bronchodilator, it can be used for the research of chronic obstructive pulmonary disease (COPD)[1].

Name	β2AR/M-receptor agonist-2

Description	β2AR/M-receptor agonist-2 (compound 15) is a muscarinic antagonist and β2 adrenoceptor agonist (MABA). β2AR/M-receptor agonist-2 shows potency to β2 adrenoceptor with an EC50 value of 3.7 nM. β2AR/M-receptor agonist-2 also has potency to human cloned M3 receptor with a Ki value of 0.73 nM. β2AR/M-receptor agonist-2 is a potent bronchodilator, it can be used for the research of chronic obstructive pulmonary disease (COPD)[1].
Related Catalog	Signaling Pathways >> Neuronal Signaling >> mAChR Research Areas >> Cardiovascular Disease Signaling Pathways >> GPCR/G Protein >> mAChR Signaling Pathways >> GPCR/G Protein >> Adrenergic Receptor Research Areas >> Inflammation/Immunology
In Vivo	β2AR/M-receptor agonist-2 剂量依赖地抑制甲基胆碱诱导的犬支气管收缩，其 ID50 值为 50 mg[1]。
References	[1]. Laura Hilton, et al. Optimized glucuronidation of dual pharmacology β-2 agonists/M3 antagonists for the treatment of COPD. MedChemComm. 2011.

Molecular Formula	C₃₆H₄₉ClN₄O₇S
Molecular Weight	717.31

The content on this webpage is sourced from various professional data sources. If you have any questions or concerns regarding the content, please feel free to contact service1@chemsrc.com.

Shanghai Nianxing Industrial Co., Ltd
China
Product Name: Palmitic acid
Price: Check
Purity: 98.0%
Delivery: 10 Day
Contact: Yang
Email: sales@echemcloud.com

β2AR/M-receptor agonist-2

Use of β2AR/M-receptor agonist-2

Names

β2AR/M-receptor agonist-2 Biological Activity

Chemical & Physical Properties

The content on this webpage is sourced from various professional data sources. If you have any questions or concerns regarding the content, please feel free to contact service1@chemsrc.com.