PPARγ/δ modulator 1
Modify Date: 2025-08-25 08:44:39
PPARγ/δ modulator 1 structure
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Common Name | PPARγ/δ modulator 1 | ||
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| CAS Number | 2089159-00-0 | Molecular Weight | 607.69 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C18H18ClIN6O3Se | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of PPARγ/δ modulator 1PPARγ/δ modulator 1 (compound 3e) is a potent PPAR modulator. PPARγ/δ modulator 1 is a PPARδ antagonist and a PPARγ partial agonist , with Ki values of 14.4 nM and 5.31 μM, respectively. PPARγ/δ modulator 1 has the EC50 of 7.3 and 12.6 μM for PPARδ corepression and adiponectin production, respectively[1]. |
| Name | PPARγ/δ modulator 1 |
|---|
| Description | PPARγ/δ modulator 1 (compound 3e) is a potent PPAR modulator. PPARγ/δ modulator 1 is a PPARδ antagonist and a PPARγ partial agonist , with Ki values of 14.4 nM and 5.31 μM, respectively. PPARγ/δ modulator 1 has the EC50 of 7.3 and 12.6 μM for PPARδ corepression and adiponectin production, respectively[1]. |
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| Related Catalog | |
| Target |
PPARδ:14.4 nM (Ki) PPARγ:5.31 μM (Ki) |
| References |
| Molecular Formula | C18H18ClIN6O3Se |
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| Molecular Weight | 607.69 |