GSK9311
Modify Date: 2024-01-02 11:36:50
GSK9311 structure
|
Common Name | GSK9311 | ||
|---|---|---|---|---|
| CAS Number | 1923851-49-3 | Molecular Weight | 437.544 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C24H31N5O3 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of GSK9311GSK9311 is a potent inhibitor of the BRPF bromodomain with pIC50 values of 6.0 and 4.3 for BRPF1 and BRPF2, respectively. |
| Name | GSK9311 |
|---|
| Description | GSK9311 is a potent inhibitor of the BRPF bromodomain with pIC50 values of 6.0 and 4.3 for BRPF1 and BRPF2, respectively. |
|---|---|
| Related Catalog | |
| Target |
IC50: 6.0 (BRPF1), 4.3 (BRPF2)[1] |
| In Vitro | GSK6853 is a potent (300 pM), soluble, cell active (20 nM), and highly selective inhibitor of the BRPF1 bromodomain, and demonstrates properties suitable for cellular and in vivo studies. GSK6853 is a less active analogue of GSK6853 in which the 5-amide is alkylated[1]. |
| References |
| Molecular Formula | C24H31N5O3 |
|---|---|
| Molecular Weight | 437.544 |