1923851-49-3
1923851-49-3 structure
- Name: GSK9311
- Chemical Name: GSK9311
- CAS Number: 1923851-49-3
- Molecular Formula: C24H31N5O3
- Molecular Weight: 437.544
- Catalog: Signaling Pathways Epigenetics Epigenetic Reader Domain
- Create Date: 2018-02-09 05:42:55
- Modify Date: 2024-01-02 11:36:50
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GSK9311 is a potent inhibitor of the BRPF bromodomain with pIC50 values of 6.0 and 4.3 for BRPF1 and BRPF2, respectively.
| Name | GSK9311 |
|---|
| Description | GSK9311 is a potent inhibitor of the BRPF bromodomain with pIC50 values of 6.0 and 4.3 for BRPF1 and BRPF2, respectively. |
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| Related Catalog | |
| Target |
IC50: 6.0 (BRPF1), 4.3 (BRPF2)[1] |
| In Vitro | GSK6853 is a potent (300 pM), soluble, cell active (20 nM), and highly selective inhibitor of the BRPF1 bromodomain, and demonstrates properties suitable for cellular and in vivo studies. GSK6853 is a less active analogue of GSK6853 in which the 5-amide is alkylated[1]. |
| References |
| Molecular Formula | C24H31N5O3 |
|---|---|
| Molecular Weight | 437.544 |