5-HT2 antagonist 1
Modify Date: 2025-08-25 22:10:54
5-HT2 antagonist 1 structure
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Common Name | 5-HT2 antagonist 1 | ||
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| CAS Number | 191592-09-3 | Molecular Weight | 400.490 | |
| Density | 1.3±0.1 g/cm3 | Boiling Point | 613.9±55.0 °C at 760 mmHg | |
| Molecular Formula | C22H29FN4O2 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | 325.1±31.5 °C | |
Use of 5-HT2 antagonist 15-HT2 antagonist 1 is a potent antagonist of 5-HT2 receptor, with weak α1 adrenoceptor blocking activity. |
| Name | 5-HT2 antagonist 1 |
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| Synonym | More Synonyms |
| Description | 5-HT2 antagonist 1 is a potent antagonist of 5-HT2 receptor, with weak α1 adrenoceptor blocking activity. |
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| Related Catalog | |
| In Vitro | 5-HT2 antagonist 1 shows 45%, 88%, 93% inhibition of 10 μM erotonin-induced contraction at 10 nM, 100 nM, 1000 nM, respectively, in guinea pig mesentcric artery. 5-HT2 antagonist 1 causes 1% and 10% inhibition of 10 μM norepinephrine-induced contraction at 10 and 100 nM, respectively, in guinea pig aorta[1]. |
| References |
| Density | 1.3±0.1 g/cm3 |
|---|---|
| Boiling Point | 613.9±55.0 °C at 760 mmHg |
| Molecular Formula | C22H29FN4O2 |
| Molecular Weight | 400.490 |
| Flash Point | 325.1±31.5 °C |
| Exact Mass | 400.227448 |
| LogP | 0.83 |
| Vapour Pressure | 0.0±1.9 mmHg at 25°C |
| Index of Refraction | 1.629 |
| 5-{3-[4-(4-Fluorophenyl)-1-piperazinyl]propyl}-8-hydroxy-1-methyl-5,6,7,8-tetrahydropyrrolo[3,2-c]azepin-4(1H)-one |
| Pyrrolo[3,2-c]azepin-4(1H)-one, 5-[3-[4-(4-fluorophenyl)-1-piperazinyl]propyl]-5,6,7,8-tetrahydro-8-hydroxy-1-methyl- |