TAK-448 acetate structure
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Common Name | TAK-448 acetate | ||
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CAS Number | 1470374-22-1 | Molecular Weight | 1285.41 | |
Density | N/A | Boiling Point | N/A | |
Molecular Formula | C60H84N16O16 | Melting Point | N/A | |
MSDS | N/A | Flash Point | N/A |
Use of TAK-448 acetateTAK-448 acetate (MVT-602 acetate) is a potent and full KISS1R agonist with an IC50 of 460 pM and an EC50 of 632 pM[1]. |
Name | TAK-448 acetate |
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Description | TAK-448 acetate (MVT-602 acetate) is a potent and full KISS1R agonist with an IC50 of 460 pM and an EC50 of 632 pM[1]. |
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Related Catalog | |
Target |
IC50: 460 pM (KISS1R)[1] EC50: 632 pM (KISS1R)[1] |
In Vivo | TAK-448 acetate (0.01-3 mg/kg; given i.h.; dosings on day 0 and 28) has greater anti-tumor effects in VCaP xenograft model[2]. Animal Model: Rat VCaP xenograft androgen-sensitive prostate cancer model (7-week-old rats) Dosage: 0.01, 0.03, 0.3, 3 mg/kg Administration: Given i.h.; dosings on day 0 and 28 Result: Had greater anti-tumor effects in VCaP xenograft model. |
References |
Molecular Formula | C60H84N16O16 |
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Molecular Weight | 1285.41 |
Storage condition | 2-8℃ |