Enzalutamide carboxylic acid
Modify Date: 2024-02-01 16:00:11
Enzalutamide carboxylic acid structure
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Common Name | Enzalutamide carboxylic acid | ||
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| CAS Number | 1242137-15-0 | Molecular Weight | 451.39400 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C20H13F4N3O3S | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of Enzalutamide carboxylic acidEnzalutamide carboxylic acid (MDV3100 carboxylic acid) is an inactive metabolite of Enzalutamide (MDV3100). Enzalutamide is an androgen receptor (AR) antagonist[1]. |
| Name | Enzalutamide Carboxylic acid |
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| Synonym | More Synonyms |
| Description | Enzalutamide carboxylic acid (MDV3100 carboxylic acid) is an inactive metabolite of Enzalutamide (MDV3100). Enzalutamide is an androgen receptor (AR) antagonist[1]. |
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| Related Catalog | |
| In Vitro | Enzalutamide is converted into its major metabolites, N-desmethyl enzalutamide and carboxylic acid enzalutamide, by cytochrome P450 (CYP) 3A4/5 and CYP2C8, respectively. N-desmethyl enzalutamide has clinically relevant anti-androgen capacities similar to enzalutamide, whereas carboxylic acid enzalutamide is inactive[1]. |
| References |
| Molecular Formula | C20H13F4N3O3S |
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| Molecular Weight | 451.39400 |
| Exact Mass | 451.06100 |
| PSA | 116.73000 |
| LogP | 4.46108 |
| Hazard Codes | Xi |
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| Enzalutamide Impurity 1 |