Enzalutamide carboxylic acid

Modify Date: 2025-08-24 20:21:25

Enzalutamide carboxylic acid Structure
Enzalutamide carboxylic acid structure
 Common Name Enzalutamide carboxylic acid
CAS Number 1242137-15-0 Molecular Weight 451.39400
Density N/A Boiling Point N/A
Molecular Formula C20H13F4N3O3S Melting Point N/A
MSDS N/A Flash Point N/A

 Use of Enzalutamide carboxylic acid


Enzalutamide carboxylic acid (MDV3100 carboxylic acid) is an inactive metabolite of Enzalutamide (MDV3100). Enzalutamide is an androgen receptor (AR) antagonist[1].

 Names

Name Enzalutamide Carboxylic acid
Synonym More Synonyms

 Enzalutamide carboxylic acid Biological Activity

Description Enzalutamide carboxylic acid (MDV3100 carboxylic acid) is an inactive metabolite of Enzalutamide (MDV3100). Enzalutamide is an androgen receptor (AR) antagonist[1].
Related Catalog
In Vitro Enzalutamide is converted into its major metabolites, N-desmethyl enzalutamide and carboxylic acid enzalutamide, by cytochrome P450 (CYP) 3A4/5 and CYP2C8, respectively. N-desmethyl enzalutamide has clinically relevant anti-androgen capacities similar to enzalutamide, whereas carboxylic acid enzalutamide is inactive[1].
References

[1]. van Nuland M, et al. Exposure-Response Assessment of Enzalutamide and Its Major Metabolites in a Real-World Cohort of Patients with Metastatic Castration-Resistant Prostate Cancer. Pharmacotherapy. 2019 Dec;39(12):1137-1145.

 Chemical & Physical Properties

Molecular Formula C20H13F4N3O3S
Molecular Weight 451.39400
Exact Mass 451.06100
PSA 116.73000
LogP 4.46108

 Safety Information

Hazard Codes Xi

 Synonyms

Enzalutamide Impurity 1
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