Sodium Channel inhibitor 1
Modify Date: 2024-01-09 19:32:46
Sodium Channel inhibitor 1 structure
|
Common Name | Sodium Channel inhibitor 1 | ||
|---|---|---|---|---|
| CAS Number | 1198117-23-5 | Molecular Weight | 473.42000 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C24H19F4N3O3 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of Sodium Channel inhibitor 1Sodium Channel inhibitor1, one of 3-Oxoisoindoline-1-carboxamides, is a novel and selective voltage-gated sodium channel for pain treatment. IC50 Value: 0.16 uM ( Na v1.7, V hold-90mV); 0.41 uM (Na v1.7, V hold-90mV) [1]Target: Na v1.7Sodium Channel inhibitor1 demonstrated concentration-dependent efficacy in preclinical behavioral pain models. |
| Name | 7-fluoro-3-oxo-2-(2-pyridin-2-ylethyl)-N-[[4-(trifluoromethoxy)phenyl]methyl]-1H-isoindole-1-carboxamide |
|---|---|
| Synonym | More Synonyms |
| Description | Sodium Channel inhibitor1, one of 3-Oxoisoindoline-1-carboxamides, is a novel and selective voltage-gated sodium channel for pain treatment. IC50 Value: 0.16 uM ( Na v1.7, V hold-90mV); 0.41 uM (Na v1.7, V hold-90mV) [1]Target: Na v1.7Sodium Channel inhibitor1 demonstrated concentration-dependent efficacy in preclinical behavioral pain models. |
|---|---|
| Related Catalog | |
| References |
| Molecular Formula | C24H19F4N3O3 |
|---|---|
| Molecular Weight | 473.42000 |
| Exact Mass | 473.13600 |
| PSA | 75.02000 |
| LogP | 4.95350 |
| Storage condition | 2-8℃ |
| FD5015 |
| Sodium Channel inhibitor 1 |