ENS-163 phosphate

Modify Date: 2024-01-09 17:18:54

ENS-163 phosphate Structure
ENS-163 phosphate structure
Common Name ENS-163 phosphate
CAS Number 117707-51-4 Molecular Weight 322.31800
Density N/A Boiling Point N/A
Molecular Formula C11H19N2O5PS Melting Point N/A
MSDS N/A Flash Point N/A

 Use of ENS-163 phosphate


ENS-163 phosphate is a selective muscarinic M1 receptor agonist.

 Names

Name (+)-(3R-cis)-3-ethyl-4,5-dihydro-4-<(1-methyl-1H-imidazol-5-yl)methyl>-2(3H)-thiophenone dihydrogen phosphate
Synonym More Synonyms

 ENS-163 phosphate Biological Activity

Description ENS-163 phosphate is a selective muscarinic M1 receptor agonist.
Related Catalog
Target

muscarinic M1 receptor[1]

In Vivo ENS-163 is a selective muscarinic M1 agonist, on long-term potentiation (LTP) is studied in a rat hippocampal slice preparation. ENS-163 facilitates the induction of long-term potentiation in rat hippocampal slices[1].
References

[1]. Boddeke EW, et al. SDZ ENS 163, a selective muscarinic M1 receptor agonist, facilitates the induction of long-term potentiation in rat hippocampal slices. Eur J Pharmacol. 1992 Nov 3;222(1):21-5.

 Chemical & Physical Properties

Molecular Formula C11H19N2O5PS
Molecular Weight 322.31800
Exact Mass 322.07500
PSA 147.76000
LogP 0.94980

 Synonyms

(3S,4R)-3-Ethyl-4-(3-methyl-3H-imidazol-4-ylmethyl)-dihydro-thiophen-2-one
compound with phosphoric acid
(+)-(3R-cis)-3-ethyl-4,5-dihydro-4-[(1-methyl-1H-imidazol-5-yl)methyl]-2(3H)-thiophenone dihydrogen phosphate
ENS-163 phosphate