- GL Biochem (Shanghai) Ltd.
- China
- Product Name: Metorphamide
- Price: $Inquiry/1g
- Purity: 98.0%
- Stocking Period: Inquiry
- Contact: Jackie Yang
- Zhejiang Hangyu API Co., Ltd
- China
- Product Name: Adrenorphin
- Price: $Inquiry/1kg
- Purity: 99.0%
- Stocking Period: 1 Day
- Contact: Vinnie
88377-68-8
88377-68-8 structure
- Name: Metorphamide
- Chemical Name: adrenorphin
- CAS Number: 88377-68-8
- Molecular Formula: C44H69N15O9S
- Molecular Weight: 984.17900
- Catalog: Peptides
- Create Date: 2018-10-13 23:23:34
- Modify Date: 2024-01-03 18:52:45
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Adrenorphin is a opioid octapeptide, acting as a potent agonist of μ-opioid receptor, with Ki of 12 nM.
| Name | adrenorphin |
|---|---|
| Synonyms |
H-TYR-GLY-GLY-PHE-MET-ARG-ARG-VAL-NH2
METORPHINAMIDE METORPHAMIDE PROENKEPHALIN (206-213) (BOVINE) adrenorphin amide TYR-GLY-GLY-PHE-MET-ARG-ARG-VAL-NH2 METORPHIN tyr-gly-gly-phe-met-arg-arg-val amide |
| Description | Adrenorphin is a opioid octapeptide, acting as a potent agonist of μ-opioid receptor, with Ki of 12 nM. |
|---|---|
| Related Catalog | |
| Target |
Ki: 12 nM (μ-opioid receptor)[1] |
| In Vitro | Adrenorphin (Metorphamide) is a opioid octapeptide from bovine brain, acts as a potent agonist of μ-opioid receptor, with Ki of 12 nM. The binding ratios of Ki for μ-opioid receptor/Ki for δ-opioid receptor of 0.04 and of Ki for μ-opioid receptor/Ki for κ-opioid receptor of 0.46[1]. Adrenorphin potently inhibits catecholamine secretion evoked by 10 μM nicotine in cultured human pheochromocytoma 6 cells, with an IC50 of 1.1 μM[2]. |
| References |
| Density | 1.42g/cm3 |
|---|---|
| Molecular Formula | C44H69N15O9S |
| Molecular Weight | 984.17900 |
| Exact Mass | 983.51200 |
| PSA | 442.14000 |
| LogP | 3.10080 |
| Index of Refraction | 1.656 |
| Storage condition | 2-8℃ |
| WGK Germany | 3 |
|---|