86434-57-3

86434-57-3 structure

Name: Beperidium iodide
Chemical Name: 4-[2-(1-Azepanyl)(1,2-benzoxazol-3-yl)acetoxy]-1-ethyl-1-methylpi peridinium iodide
CAS Number: 86434-57-3
Molecular Formula: C₂₃H₃₄IN₃O₃
Molecular Weight: 527.43900
Catalog: Signaling Pathways GPCR/G Protein mAChR
Create Date: 2017-10-04 01:18:29
Modify Date: 2024-01-11 11:02:00
Beperidium iodide shows a competitive antagonistic effect against acetylcholine receptor with a pA2 of 7.93.

Name	4-[2-(1-Azepanyl)(1,2-benzoxazol-3-yl)acetoxy]-1-ethyl-1-methylpi peridinium iodide
Synonyms	4-<2-(1,2-benzisoxazol-3-yl)-2-(hexahydro-1H-azepin-1-yl)acetoxy>-1-ethyl-1-methylpiperidinium iodide 3-(5-tert-butyl-isoxazol-3-yl)-1-ethyl-1-methyl-urea Urea,N'-[5-(1,1-dimethylethyl)-3-isoxazolyl]-N-ethyl-N-methyl 1-ethyl-1-methyl-3-(5-t-butyl-3-isoxazolyl)urea 1-ethyl-1-methyl-4-[2-hexamethyleneimino-2-(1,2-benzisoxazol-3-yl)acetoxy]piperidinium iodide Beperidium iodide

Description	Beperidium iodide shows a competitive antagonistic effect against acetylcholine receptor with a pA2 of 7.93.
Related Catalog	Signaling Pathways >> GPCR/G Protein >> mAChR Signaling Pathways >> Neuronal Signaling >> mAChR Research Areas >> Inflammation/Immunology
Target	pA2: 7.93 (Acetylcholine receptor)[1]
References	[1]. Kawashima K, et al. Pharmacological properties of the novel antimuscarinic agent 4-[2-(1,2-benzisoxazol-3-yl)-2-(hexahydro-1H-azepin-1-yl)a cetoxy]-1-et hyl-1- methylpiperidinium iodide. Arzneimittelforschung. 1986 Jun;36(6):927-35.