Name | 6-(4-methylpiperazin-1-yl)-11H-benzo[c][1]benzazepine |
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Synonyms |
6-(4-Methyl-1-piperazinyl)morphanthridine
Perlapina [Spanish] Perlapinum [INN-Latin] 6-(4-Methyl-1-piperazinyl)-morphanthridin Hypnodin AW-14'2333 6-(4-methyl-piperazin-1-yl)-11H-dibenzo[b,e]azepine Morphanthridine,6-(4-methyl-1-piperazinyl) Perlapin Perlapina [INN-Spanish] MP-11 6-(4-Methyl-piperazin-1-yl)-morphanthridin PERLAPINE |
Description | Perlapine is a potent muscarinic DREADD (Designer Receptors Exclusively Activated by Designer Drugs) agonist Perlapine exhibits >10000-fold selectivity for hM3Dq over hM3 receptors[1]. |
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Related Catalog | |
References |
Molecular Formula | C19H21N3 |
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Molecular Weight | 291.39000 |
Exact Mass | 291.17400 |
PSA | 18.84000 |
LogP | 2.22790 |
Vapour Pressure | 7.74E-08mmHg at 25°C |
CHEMICAL IDENTIFICATION
HEALTH HAZARD DATAACUTE TOXICITY DATA
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~% 1977-11-3 |
Literature: Sinha, Ashok Kumar; Nizamuddin, S. Indian Journal of Chemistry, Section B: Organic Chemistry Including Medicinal Chemistry, 1984 , vol. 23, # 2 p. 165 |
~% 1977-11-3 |
Literature: Sinha, Ashok Kumar; Nizamuddin, S. Indian Journal of Chemistry, Section B: Organic Chemistry Including Medicinal Chemistry, 1984 , vol. 23, # 2 p. 165 |
~% 1977-11-3 |
Literature: Sinha, Ashok Kumar; Nizamuddin, S. Indian Journal of Chemistry, Section B: Organic Chemistry Including Medicinal Chemistry, 1984 , vol. 23, # 2 p. 165 |
~% 1977-11-3 |
Literature: Sinha, Ashok Kumar; Nizamuddin, S. Indian Journal of Chemistry, Section B: Organic Chemistry Including Medicinal Chemistry, 1984 , vol. 23, # 2 p. 165 |
Precursor 4 | |
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DownStream 0 |