Name | α-Helical CRF(9-41) |
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Description | α-Helical CRF(9-41) is a competitive CRF2 receptor antagonist with KB of ~100 nM. α-Helical CRF(9-41) is also a partial agonist of CRF1 receptor with an EC50 of 140 nM[1][2]. |
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Related Catalog | |
Target |
KB: ~100 nM (CRF2 receptor)[2] EC50: 140 nM (CRF1 receptor)[2] |
References |
Molecular Formula | C166H274N46O53S2 |
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Molecular Weight | 3826.40 |