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Product Name: OMDM-3
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616884-64-1

616884-64-1 structure

616884-64-1 structure

Name: OMDM-3
Chemical Name: OMDM-3
CAS Number: 616884-64-1
Molecular Formula: C₂₉H₄₃NO₃
Molecular Weight: 453.66
Catalog: Research Areas Neurological Disease
Create Date: 2020-06-01 19:45:27
Modify Date: 2024-01-09 18:38:24
OMDM-3 is a selective and metabolically stable inhibitor of anandamide cellular uptake (ACU), with a Ki of 16.6 μM[1].

Name	OMDM-3

Description	OMDM-3 is a selective and metabolically stable inhibitor of anandamide cellular uptake (ACU), with a Ki of 16.6 μM[1].
Related Catalog	Research Areas >> Neurological Disease
Target	Ki: 16.6 μM (anandamide cellular uptake)[1]
In Vitro	OMDM-3 shows poor affinity for either CB1 (Ki=6.1 μM) or CB2 (Ki>10 μM) receptors in rat brain and spleen membranes, respectively. OMDM-3 has almost no activity at vanilloid receptors in the intracellular calcium assay carried out with intact cells over-expressing the human VR1 (EC50>10 μM), and no activity as inhibitors of FAAH in N18TG2 cell membranes (Ki>50 μM)[1].
References	[1]. Ortar G, et al. Novel selective and metabolically stable inhibitors of anandamide cellular uptake. Biochem Pharmacol. 2003 May 1;65(9):1473-81.

Molecular Formula	C₂₉H₄₃NO₃
Molecular Weight	453.66

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