2173153-38-1
2173153-38-1 structure
- Name: BMS-212
- Chemical Name: BMS-212
- CAS Number: 2173153-38-1
- Molecular Formula: C25H30N3O9PS2
- Molecular Weight: 611.621
- Create Date: 2020-01-11 21:20:50
- Modify Date: 2025-08-28 10:47:11
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BMS-212 is a potent and selective stimulator of glucokinase (GK) (EC50 = 35 nM) that is promisingly used as an antidiabetic.
| Name | BMS-212 |
|---|
| Description | BMS-212 is a potent and selective stimulator of glucokinase (GK) (EC50 = 35 nM) that is promisingly used as an antidiabetic. |
|---|---|
| In Vitro | BMS-212 is a potent and selective stimulator of glucokinase (GK) (EC50 = 35 nM) that is promisingly used as an antidiabetic. BMS-212 has a preference for GK in liver over GK in pancreas, of which the activation may lead to non-glucose-dependent insulin secretion. Half-life of BMS-212 is 4.2h, and oral bioavailability is 15%. |
| Molecular Formula | C25H30N3O9PS2 |
|---|---|
| Molecular Weight | 611.621 |