2101951-67-9
2101951-67-9 structure
- Name: LSD1-IN-11p
- Chemical Name: LSD1-IN-11p
- CAS Number: 2101951-67-9
- Molecular Formula: C22H24N6O3
- Molecular Weight: 420.473
- Create Date: 2020-01-11 20:34:51
- Modify Date: 2024-04-05 11:55:17
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LSD1-IN-11p is a reversible LSD1 inhibitor with IC50/Kd of 79/21 nM; upregulates the expression of the surrogate cellular biomarker CD86 (IC50=0.52 uM); has moderate oral bioavailability in mice (F%=38%).
| Name | LSD1-IN-11p |
|---|
| Description | LSD1-IN-11p is a reversible LSD1 inhibitor with IC50/Kd of 79/21 nM; upregulates the expression of the surrogate cellular biomarker CD86 (IC50=0.52 uM); has moderate oral bioavailability in mice (F%=38%). |
|---|---|
| References | References 1. Mould DP, et al. Bioorg Med Chem Lett. 2017 Jul 15;27(14):3190-3195. View Related Products by Target Histone Demethylase |
| Molecular Formula | C22H24N6O3 |
|---|---|
| Molecular Weight | 420.473 |