1663564-42-8
1663564-42-8 structure
- Name: GAT-100
- Chemical Name: GAT100
- CAS Number: 1663564-42-8
- Molecular Formula: C25H28N4OS
- Molecular Weight: 432.581
- Create Date: 2018-06-26 03:54:17
- Modify Date: 2025-08-25 22:38:02
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GAT-100 (GAT100) is a potent, selective CB1R negative allosteric modulator (NAM) with cAMP EC50 and β-arr EC50 of 174 nM and 2.1 nM, does not exhibit inverse agonism.
| Name | GAT100 |
|---|---|
| Synonyms |
GAT100
Thiocyanic acid, 3-ethyl-2-[[[2-[4-(1-piperidinyl)phenyl]ethyl]amino]carbonyl]-1H-indol-5-yl ester 3-Ethyl-2-({2-[4-(1-piperidinyl)phenyl]ethyl}carbamoyl)-1H-indol-5-yl thiocyanate |
| Density | 1.3±0.1 g/cm3 |
|---|---|
| Boiling Point | 716.3±60.0 °C at 760 mmHg |
| Molecular Formula | C25H28N4OS |
| Molecular Weight | 432.581 |
| Flash Point | 387.0±32.9 °C |
| Exact Mass | 432.198395 |
| LogP | 5.90 |
| Vapour Pressure | 0.0±2.3 mmHg at 25°C |
| Index of Refraction | 1.671 |