AT-121 hydrochloride
Names
[ CAS No. ]:
2099681-71-5
[ Name ]:
AT-121 hydrochloride
Biological Activity
[Description]:
AT-121 hydrochloride is a bifunctional nociception and mu opioid receptor agonist, with Kis of 3.67 and 16.49 nM, respectively. AT-121 hydrochloride is a safe, non-addictive analgesic, and shows antinociceptive and antiallodynic effects[1].
[Related Catalog]:
[In Vivo]
AT-121 hydrochloride (0.003-0.03 mg/kg; s.c.) produces potent antinociceptive effect[1]. Animal Model: Adult male and female rhesus monkeys[1] Dosage: 0.003-0.03 mg/kg Administration: Subcutaneous Result: Produced antinociceptive effects against an acute noxious stimulus, 50 °C water, in a dose-dependent.
[References]
Chemical & Physical Properties
[ Molecular Formula ]:
C24H39ClN4O3S
[ Molecular Weight ]:
499.11