Herkinorin

Names

[ CAS No. ]:
862073-77-6

[ Name ]:
Herkinorin

[Synonym ]:
BF3DNCA methyl ester
herkinorin

Biological Activity

[Description]:

Herkinorin is a potent and selective agonist of µ opioid receptor with a Ki of 45 nM Herkinorin is widely used for pain research[1].

[Related Catalog]:

Signaling Pathways >> GPCR/G Protein >> Opioid Receptor

Signaling Pathways >> Neuronal Signaling >> Opioid Receptor

Research Areas >> Neurological Disease

[References]

[1]. Lamb K, et al. Antinociceptive effects of herkinorin, a MOP receptor agonist derived from salvinorin A in the formalin test in rats: new concepts in mu opioid receptor pharmacology: from a symposium on new concepts in mu-opioid pharmacology. Drug Alcohol Depend. 2012 Mar 1;121(3):181-8.

Chemical & Physical Properties

[ Molecular Formula ]:
C₂₈H₃₀O₈

[ Molecular Weight ]:
494.53300

[ Exact Mass ]:
494.19400

[ PSA ]:
109.11000

[ LogP ]:
4.29400

Related Compounds

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