GSK215083

Names

[ Name ]:
GSK215083

[Synonym ]:
unii-8gfe8j4n0z

Biological Activity

[Description]:

GSK215083 is a high affinity 5-HT6 receptor antagonist. GSK215083 can serves as a promising 5-HT6 radioligand candidate by radiolabeled with (11)C via methylation[1].

[Related Catalog]:

Research Areas >> Others

Signaling Pathways >> GPCR/G Protein >> 5-HT Receptor

Signaling Pathways >> Neuronal Signaling >> 5-HT Receptor

[Target]

5-HT6 Receptor

[References]

[1]. Parker CA, et al. Radiosynthesis and characterization of 11C-GSK215083 as a PET radioligand for the 5-HT6 receptor. J Nucl Med. 2012 Feb;53(2):295-303.

Chemical & Physical Properties

[ Molecular Formula ]:
C₂₀H₂₀FN₃O₂S

[ Molecular Weight ]:
385.46

[ Exact Mass ]:
385.12600

[ PSA ]:
61.89000

[ LogP ]:
4.04220

Related Compounds

The content on this webpage is sourced from various professional data sources. If you have any questions or concerns regarding the content, please feel free to contact service1@chemsrc.com.