M1/M4 muscarinic agonist 3

Names

[ CAS No. ]:
2640109-30-2

[ Name ]:
M1/M4 muscarinic agonist 3

Biological Activity

[Description]:

M1/M4 muscarinic agonist 3 (compound 44) is a muscarinic mAChR M1/M4 agonist with EC50s of 31 nM and 9.3 nM, respectively[1].

[Related Catalog]:

Signaling Pathways >> Neuronal Signaling >> mAChR
Signaling Pathways >> GPCR/G Protein >> mAChR
Research Areas >> Neurological Disease

[Target]

EC50: 31 nM (M1 muscarinic receptor), 9.3 nM (M4 muscarinic receptor)[1]


[References]

[1]. Thomson C G et al. Transaminases Provide Key Chiral Building Blocks for the Synthesis of Selective M1/M4 Agonists[J]. ACS Medicinal Chemistry Letters, 2023.

Chemical & Physical Properties

[ Molecular Formula ]:
C23H31FN2O3

[ Molecular Weight ]:
402.50

Related Compounds

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