CB1R Allosteric modulator 2

Names

[ CAS No. ]:
2513102-64-0

[ Name ]:
CB1R Allosteric modulator 2

Biological Activity

[Description]:

CB1R Allosteric modulator 2 (compound 18) is a potent CB1R allosteric modulator. CB1R Allosteric modulator 2 shows negatively affects the functional activity of orthosteric ligands (NAM) at CB1Rs[1].

[Related Catalog]:

Research Areas >> Others
Signaling Pathways >> GPCR/G Protein >> Cannabinoid Receptor

[Target]

hCB1-R


[References]

[1]. Meini S,et al. PSNCBAM-1 analogs: Structural evolutions and allosteric properties at cannabinoid CB1 receptor. Eur J Med Chem. 2020 Oct 1;203:112606.

Chemical & Physical Properties

[ Molecular Formula ]:
C19H15ClFN3O

[ Molecular Weight ]:
355.79

Related Compounds