μ opioid receptor agonist 3

Names

[ CAS No. ]:
2378397-91-0

[ Name ]:
μ opioid receptor agonist 3

Biological Activity

[Description]:

μ opioid receptor agonist 3 (compound 20) is a potent μ opioid receptor (µOR) agonist with an EC50 of 0.87 nM. μ opioid receptor agonist 3 has the potential for pain and neuropsychiatric indications research[1].

[Related Catalog]:

Signaling Pathways >> GPCR/G Protein >> Opioid Receptor
Signaling Pathways >> Neuronal Signaling >> Opioid Receptor
Research Areas >> Neurological Disease

[Target]

μ Opioid Receptor/MOR:0.82 nM (EC50)


[References]

[1]. Alok Nerurkar, et al. Novel series of tunable µOR modulators with enhanced brain penetration for the treatment of opioid use disorder, pain and neuropsychiatric indications. Bioorg Med Chem Lett. 2023 Aug 15:92:129405.  

Chemical & Physical Properties

[ Molecular Formula ]:
C22H28N2O2

[ Molecular Weight ]:
352.47

Related Compounds

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