EHMT2-IN-1

Names

[ Name ]:
EHMT2-IN-1

Biological Activity

[Description]:

EHMT2-IN-1 is a potent EHMT inhibitor, with IC50s of all <100 nM for EHMT1 peptide, EHMT2 peptide and cellular EHMT2. Used in the research of blood disorder or cancer[1].

[Related Catalog]:

Research Areas >> Cancer

Signaling Pathways >> Epigenetics >> Histone Methyltransferase

[Target]

EHMTI PEP:<100 nM (IC50)

EHMT2 PEP:<100 nM (IC50)

EHMT2 ICW:<100 nM (IC50)

[In Vitro]

EHMT2-IN-1 (Compound 108) potent EHMT inhibitor, with IC50s of all <100 nM for EHMT1 peptide, EHMT2 peptide and cellular EHMT2[1].

[References]

[1]. John Emmerson Campbell, et al. Amine-substituted heterocyclic compounds as ehmt2 inhibitors and methods of use thereof. WO2018118842A1

Chemical & Physical Properties

[ Molecular Formula ]:
C₁₈H₂₃N₇O

[ Molecular Weight ]:
353.42

[ Storage condition ]:
2-8℃

Related Compounds

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