2230849-55-3

2230849-55-3 structure

Name: EHMT2-IN-1
Chemical Name: EHMT2-IN-1
CAS Number: 2230849-55-3
Molecular Formula: C₁₈H₂₃N₇O
Molecular Weight: 353.42
Catalog: Signaling Pathways Epigenetics Histone Methyltransferase
Create Date: 2019-06-01 16:10:31
Modify Date: 2025-08-27 13:02:11
EHMT2-IN-1 is a potent EHMT inhibitor, with IC50s of all <100 nM for EHMT1 peptide, EHMT2 peptide and cellular EHMT2. Used in the research of blood disorder or cancer[1].

Name	EHMT2-IN-1

Description	EHMT2-IN-1 is a potent EHMT inhibitor, with IC50s of all <100 nM for EHMT1 peptide, EHMT2 peptide and cellular EHMT2. Used in the research of blood disorder or cancer[1].
Related Catalog	Research Areas >> Cancer Signaling Pathways >> Epigenetics >> Histone Methyltransferase
Target	EHMTI PEP:<100 nM (IC50) EHMT2 PEP:<100 nM (IC50) EHMT2 ICW:<100 nM (IC50)
In Vitro	EHMT2-IN-1 (Compound 108) potent EHMT inhibitor, with IC50s of all <100 nM for EHMT1 peptide, EHMT2 peptide and cellular EHMT2[1].
References	[1]. John Emmerson Campbell, et al. Amine-substituted heterocyclic compounds as ehmt2 inhibitors and methods of use thereof. WO2018118842A1