AZ-8838

Names

[ Name ]:
AZ-8838

[Description]:

AZ-8838 (AZ8838) is a potent, and selective PAR2 antagonist with Kd of 125 nM; shows excellent selectivity over PAR1 and PAR4 (>50 uM).

[References]

References 1. Cheng RKY, et al. Nature. 2017 May 4;545(7652):112-115. View Related Products by Target Protease-activated Receptor (PAR)

[ Molecular Formula ]:
C₁₃H₁₅FN₂O

[ Molecular Weight ]:
234.274