SMYD3-IN-1

Names

[ CAS No. ]:
2095160-79-3

[ Name ]:
SMYD3-IN-1

Biological Activity

[Description]:

SMYD3-IN-1 (compound 29) is an irreversible and selective inhibitor of SMYD3 (SET and MYND domain containing 3), with an IC50 of 11.7 nM[1].

[Related Catalog]:

Signaling Pathways >> Epigenetics >> Histone Methyltransferase

Research Areas >> Others

[Target]

SMYD3:11.7 nM (IC50)

[References]

[1]. Huang C, et al. Discovery of Irreversible Inhibitors Targeting Histone Methyltransferase, SMYD3. ACS Med Chem Lett. 2019 May 23;10(6):978-984.

Chemical & Physical Properties

[ Molecular Formula ]:
C₂₈H₃₁ClN₄O₃

[ Molecular Weight ]:
507.02

Related Compounds

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