CYN 154806

Names

[ Name ]:
CYN 154806

Biological Activity

[Description]:

CYN 154806, a cyclic octapeptide, is a potent and selective somatostatin sst2 receptor antagonist, with pIC50 values of 8.58, 5.41, 6.07, 5.76 and 6.48 for human recombinant sst2, sst1, sst3, sst4 and sst5 receptors respectively[1][2].

[Related Catalog]:

Signaling Pathways >> GPCR/G Protein >> Somatostatin Receptor

Research Areas >> Others

[Target]

Somatostatin Receptor[1].

[References]

[1]. Bass RT, et al. Identification and characterization of novel somatostatin antagonists. Mol Pharmacol. 1996 Oct;50(4):709-15.

[2]. Feniuk W, et al. Selective somatostatin sst(2) receptor blockade with the novel cyclic octapeptide, CYN-154806. Neuropharmacology. 2000 Jun 8;39(8):1443-50.

Chemical & Physical Properties

[ Molecular Formula ]:
C₅₆H₆₈N₁₂O₁₄S₂

[ Molecular Weight ]:
1197.34

[ Exact Mass ]:
1196.44000

[ PSA ]:
474.81000

[ LogP ]:
4.78680

MSDS

Click to get detail MSDS

Related Compounds

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