183658-72-2

183658-72-2 structure

Name: CYN 154806
Chemical Name: cyn 154806
CAS Number: 183658-72-2
Molecular Formula: C₅₆H₆₈N₁₂O₁₄S₂
Molecular Weight: 1197.34
Catalog: Signaling Pathways GPCR/G Protein Somatostatin Receptor
Create Date: 2017-10-15 07:47:44
Modify Date: 2024-01-10 18:56:07
CYN 154806, a cyclic octapeptide, is a potent and selective somatostatin sst2 receptor antagonist, with pIC50 values of 8.58, 5.41, 6.07, 5.76 and 6.48 for human recombinant sst2, sst1, sst3, sst4 and sst5 receptors respectively[1][2].

Name	cyn 154806

Description	CYN 154806, a cyclic octapeptide, is a potent and selective somatostatin sst2 receptor antagonist, with pIC50 values of 8.58, 5.41, 6.07, 5.76 and 6.48 for human recombinant sst2, sst1, sst3, sst4 and sst5 receptors respectively[1][2].
Related Catalog	Signaling Pathways >> GPCR/G Protein >> Somatostatin Receptor Research Areas >> Others
Target	Somatostatin Receptor[1].
References	[1]. Bass RT, et al. Identification and characterization of novel somatostatin antagonists. Mol Pharmacol. 1996 Oct;50(4):709-15. [2]. Feniuk W, et al. Selective somatostatin sst(2) receptor blockade with the novel cyclic octapeptide, CYN-154806. Neuropharmacology. 2000 Jun 8;39(8):1443-50.