CK1-IN-1

Names

[ Name ]:
CK1-IN-1

Biological Activity

[Description]:

CK1-IN-1 is a casein kinase 1 (CK1) inhibitor extracted from patent WO2015119579A1, compound 1c, has IC50s of 15 nM, 16 nM, 73 nM for CK1δ, and CK1ε, p38σ MAPK, respectively[1].

[Related Catalog]:

Research Areas >> Inflammation/Immunology

Signaling Pathways >> Cell Cycle/DNA Damage >> Casein Kinase

Signaling Pathways >> Stem Cell/Wnt >> Casein Kinase

[Target]

CKIδ:15 nM (IC50)

CK1ϵ:16 nM (IC50)

[References]

[1]. Filip LACO,et al. 2,4,5-tri-substituted azole-based casein kinase 1 inhibitors as inducers for cardiomyogenesis. WO2015119579A1.

Chemical & Physical Properties

[ Molecular Formula ]:
C₂₄H₁₅F₂N₃

[ Molecular Weight ]:
383.39

Related Compounds

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