5-HT2A&5-HT2C agonist-1

Names

[ CAS No. ]:
1640-02-4

[ Name ]:
5-HT2A&5-HT2C agonist-1

Biological Activity

[Description]:

5-HT2A&5-HT2C agonist-1 (Example 2) is a 5-HT2A & 5-HT2C agonist, with IC50s of 196 nM and 0.9 nM respectively. 5-HT2A&5-HT2C agonist-1 can be used for research of depression, alcoholism, tobacco and cocaine addiction, inflammation, cluster headache, PTSD, seizure disorders and other CNS disorders[1].

[Related Catalog]:

Research Areas >> Cancer
Research Areas >> Inflammation/Immunology
Research Areas >> Neurological Disease
Signaling Pathways >> GPCR/G Protein >> 5-HT Receptor
Signaling Pathways >> Neuronal Signaling >> 5-HT Receptor

[Target]

196 nM and 0.9 nM (5-HT2A&5-HT2C)[1]


[References]

[1]. Alan Kozikowski, et al. 3-(2-(aminoethyl)-indol-4-ol derivatives, methods of preparation thereof, and the use as 5-ht2 receptor modulators. Patent. WO2021179091.

Chemical & Physical Properties

[ Molecular Formula ]:
C14H20N2O

[ Molecular Weight ]:
232.32


Related Compounds

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