CDK8-IN-4

Names

[ CAS No. ]:
1613638-82-6

[ Name ]:
CDK8-IN-4

Biological Activity

[Description]:

CDK8-IN-4 is an inhibitor of CDK8 extracted from patent WO2014090692A1, compound example 16, with an IC50 of 0.2 nM.

[Related Catalog]:

Research Areas >> Cancer

[Target]

IC50: 0.2 nM (CDK8)[1]


[References]

[1]. Cheng Z, et al. Novel bi-ring phenyl-pyridines/pyrazines for the treatment of cancer. WO2014090692A1


[Related Small Molecules]

Abemaciclib(LY2835219) | Ribociclib (LEE011) | Dinaciclib (SCH727965) | THZ1 2HCl | Roscovitine (CYC202) | THZ531 | RO-3306 | Flavopiridol | NVP 2 | BAY-1143572 Racemate | CYC-065 | AZD5438 | BIO | Kenpaullone | SNS-032 (BMS-387032)

Chemical & Physical Properties

[ Molecular Formula ]:
C20H18N4O

[ Molecular Weight ]:
330.38

Related Compounds