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AEF0117

Names

[ CAS No. ]:
1610878-71-1

[ Name ]:
AEF0117

Biological Activity

[Description]:

AEF0117 a signaling-specific inhibitor of the cannabinoid receptor 1 (CB1-SSi). AEF0117 plays an important role in Cannabis use disorder (CUD)[1].

[Related Catalog]:

Research Areas >> Neurological Disease
Signaling Pathways >> GPCR/G Protein >> Cannabinoid Receptor

[Target]

cannabinoid receptor 1 (CB1-SSi)[1]


[References]

[1]. Margaret Haney, et al. Signaling-specific inhibition of the CB1 receptor for cannabis use disorder: phase 1 and phase 2a randomized trials. Nat Med. 2023 Jun;29(6):1487-1499.  

Chemical & Physical Properties

[ Molecular Formula ]:
C29H40O3

[ Molecular Weight ]:
436.63


Related Compounds