(R)-PQ-912

Names

[ CAS No. ]:
1276021-64-7

[ Name ]:
(R)-PQ-912

Biological Activity

[Description]:

(R)-PQ-912 is a glutaminyl cyclase (QC) inhibitor extracted from patent WO2011029920A1, example 13, has an IC50 of 30.2 μM and a Ki of 7.25 μM for hQC[1].

[Related Catalog]:

Signaling Pathways >> Others >> Others
Research Areas >> Neurological Disease

[References]

[1]. Ulrich Heiser, et al. Heterocylcic derivatives as inhibitors of glutaminyl cyclase.

Chemical & Physical Properties

[ Molecular Formula ]:
C19H20N4O2

[ Molecular Weight ]:
336.39

Related Compounds