Rac-PQ-912

Names

[ CAS No. ]:
1276021-63-6

[ Name ]:
Rac-PQ-912

Biological Activity

[Description]:

Rac-PQ-912 is a glutaminyl cyclase (QC) inhibitor extracted from patent WO2011029920A1, compound example 12, has an EC50 of 482 nM and a Ki of 62.5 nM for hQC[1].

[Related Catalog]:

Research Areas >> Others

[Target]

EC50: 482 nM (hQC) Ki: 62.5 nM (hQC)[1]


[References]

[1]. Ulrich Heiser, et al. Heterocylcic derivatives as inhibitors of glutaminyl cyclase.

Chemical & Physical Properties

[ Molecular Formula ]:
C19H20N4O2

[ Molecular Weight ]:
336.39

Related Compounds