Epoxidation of flavones by dimethyldioxirane

W Adam, D Golsch, L Hadjiarapoglou…

Index: Adam, Waldemar; Golsch, Dieter; Hadjiarapoglou, Lazaros Journal of Organic Chemistry, 1991 , vol. 56, # 26 p. 7292 - 7297

Full Text: HTML

Citation Number: 43

Abstract

The synthesis of epoxides 2 by epoxidation of flavones 1 with isolated dimethyldioxirane (as acetone solution) at subambient temperatures is reported. These labile epoxides were isolated and completely characterized by UV, IR,'H and I3C NMR, MS, and C, H analyses. Warming to room temperature led to rearrangement to afford quantitatively the 3- hydroxyflavones Sb, h, i, n. Treatment of the epoxides 2b, f with methanol led to the 3- ...

Related Articles:

Regioselective synthesis of flavone derivatives via DMAP-catalyzed cyclization of o-alkynoylphenols

[Yoshida, Masahito; Fujino, Yuta; Saito, Koya; Doi, Takayuki Tetrahedron, 2011 , vol. 67, # 51 p. 9993 - 9997]

K2CO3-Catalyzed Synthesis of Chromones and 4-Quinolones through the Cleavage of Aromatic C–O Bonds

[Zhao, Jie; Zhao, Yufen; Fu, Hua Organic Letters, 2012 , vol. 14, # 11 p. 2710 - 2713]

Synthesis of Chromones through LiOtBu/Air??Mediated Oxidation and Regioselective Cyclization of o??Hydroxyphenyl Propargyl Carbinols

[Zhang, Shuai; Wan, Changfeng; Wang, Qiang; Zhang, Baiqun; Gao, Lingfeng; Zha, Zhenggen; Wang, Zhiyong European Journal of Organic Chemistry, 2013 , # 11 p. 2080 - 2083]

Ionic liquid mediated Cu-catalyzed cascade oxa-Michael-oxidation: efficient synthesis of flavones under mild reaction conditions

[Du, Zhiyun; Ng, Huifen; Zhang, Kun; Zeng, Huaqiang; Wang, Jian Organic and Biomolecular Chemistry, 2011 , vol. 9, # 20 p. 6930 - 6933]

Palladium??Catalyzed Carbonylation Reaction of Aryl Bromides with 2??Hydroxyacetophenones to Form Flavones

[Wu, Xiao-Feng; Neumann, Helfried; Beller, Matthias Chemistry - A European Journal, 2012 , vol. 18, # 40 p. 12595 - 12598]

More Articles...