β-Selective C-arylation of silyl protected 1, 6-anhydroglucose with arylalanes: the synthesis of SGLT2 inhibitors

JP Henschke, PY Wu, CW Lin, SF Chen…

Index: Miyoshi, Tetsuya; Matsuya, Syota; Tsugawa, Mikako; Sato, Shohei; Ueda, Masafumi; Miyata, Okiko Organic Letters, 2013 , vol. 15, # 13 p. 3374 - 3377

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Abstract

... Volume: Page: ... and cross-couplings.(13) The relatively high Lewis acidity of the aluminum centers combined with nucleophilic organic ligands renders ... as synthetic reagents on their own.(14) For example, in related work, Yamamoto et al.(15) demonstrated the ...

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