Tetrahedron letters

rel-(1R, 4R, 5S)-5-hydroxy-3-oxo-2-azabicyclo [2.2. 0] hexane, a stable synthetic equivalent of 4-(2-oxoethyl) azetidin-2-one

N Katagiri, M Sato, T Naito, M Muto, T Sakamoto…

Index: Katagiri, Nobuya; Sato, Masayuki; Naito, Toshihiko; Muto, Makoto; Sakamoto, Toshiyuki; et al. Tetrahedron Letters, 1984 , vol. 25, # 49 p. 5665 - 5668

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Abstract

Download full text in PDF Opens in a new window. Article suggestions will be shown in a dialog on return to ScienceDirect. ... Please enable JavaScript to use all the features on this page. ... The title compound, a synthetic equivalent of 4-(2-oxoethyl)-azetidin-2-one, has been synthesized as a stable crystalline solid either from 4-( -butyldimethylsilyloxy)- or 4-benzyloxy-2-pyridone photopyridone formation, catalytic hydrogenation, and deblocking of the protecting group.

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