Helvetica chimica acta

First Use of Benzyl Phosphites in the Michaelis??Arbuzov Reaction synthesis of mono??, Di??, and triphosphate analogs

M Saady, L Lebeau, C Mioskowski

Index: Saady, Mourad; Lebeau, Luc; Mioskowski, Charles Helvetica Chimica Acta, 1995 , vol. 78, p. 670 - 678

Full Text: HTML

Citation Number: 39

Abstract

Abstract Benzyl phosphites were used in the Micaelis-Arbuzov reaction. Special experimental conditions allowed preparation of a set of phosphonate analogs of mono-, di-, and triphosphate. Furthermore, regioselective monodeprotection makes these molecules useful building blocks for the synthesis of analogs of polyphosphorylated compounds of biological interest (eg nucleotides), after removal of all phosphonate benzyl ester groups ...

Related Articles:

Mild and efficient Cs 2 CO 3-promoted synthesis of phosphonates

[Cohen, Richard J.; Fox, Daniel L.; Eubank, Jarrod F.; Salvatore, Ralph Nicholas Tetrahedron Letters, 2003 , vol. 44, # 47 p. 8617 - 8621]

Tailoring the Specificity and Reactivity of a Mechanism??Based Inactivator of Glucocerebrosidase for Potential Therapeutic Applications

[Rempel, Brian P.; Tropak, Michael B.; Mahuran, Don J.; Withers, Stephen G. Angewandte Chemie - International Edition, 2011 , vol. 50, # 44 p. 10381 - 10383]

More Articles...