Sigma-2 Radioligand 1
Modify Date: 2024-01-13 20:43:51
Sigma-2 Radioligand 1 structure
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Common Name | Sigma-2 Radioligand 1 | ||
|---|---|---|---|---|
| CAS Number | 2860554-32-9 | Molecular Weight | 427.51 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C24H30FN3O3 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of Sigma-2 Radioligand 1Sigma-2 Radioligand 1 (compound 1) is a Sigma-2 selective ligand. Sigma-2 Radioligand 1 has good biodistribution in mice and good in vivo activity in rats. [18F] Modified Sigma-2 Radioligand 1 for visualization of tumors in micro-PET/CT imaging, exhibiting high tumor uptake and tumor-to-background ratio. Experiments show that Sigma-2 Radioligand 1 binds highly specifically in U87MG glioma xenografts[1]. |
| Name | Sigma-2 Radioligand 1 |
|---|
| Description | Sigma-2 Radioligand 1 (compound 1) is a Sigma-2 selective ligand. Sigma-2 Radioligand 1 has good biodistribution in mice and good in vivo activity in rats. [18F] Modified Sigma-2 Radioligand 1 for visualization of tumors in micro-PET/CT imaging, exhibiting high tumor uptake and tumor-to-background ratio. Experiments show that Sigma-2 Radioligand 1 binds highly specifically in U87MG glioma xenografts[1]. |
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| Related Catalog | |
| Target |
Ki: 2.57 nM (Sigma-2, σ2)[1] |
| References |
| Molecular Formula | C24H30FN3O3 |
|---|---|
| Molecular Weight | 427.51 |