PKM2 activator 3
Modify Date: 2025-08-26 21:52:24
PKM2 activator 3 structure
|
Common Name | PKM2 activator 3 | ||
|---|---|---|---|---|
| CAS Number | 1346113-84-5 | Molecular Weight | 372.77 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C15H11ClF2N2O3S | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of PKM2 activator 3PKM2 activator 3 is a potent PKM2 activator with an AC50 value of 90 nM. PKM2 activator 3 has good Caco-2 permeability, a low efflux ratio and high microsomal stability. PKM2 activator 3 can be used for researching anticancer[1]. (AC50: the concentration which gives 50% activation of enzyme.) |
| Name | PKM2 activator 3 |
|---|
| Description | PKM2 activator 3 is a potent PKM2 activator with an AC50 value of 90 nM. PKM2 activator 3 has good Caco-2 permeability, a low efflux ratio and high microsomal stability. PKM2 activator 3 can be used for researching anticancer[1]. (AC50: the concentration which gives 50% activation of enzyme.) |
|---|---|
| Related Catalog | |
| Target |
PKM2[1] |
| In Vivo | PKM2 activator 3 (compound 66) has good Caco-2 permeability, a low efflux ratio (0.84) and high microsomal stability (t1/2 = 277.2 min in human liver microsomes and 117.5 min in mouse liver microsomes)[1]. |
| References |
| Molecular Formula | C15H11ClF2N2O3S |
|---|---|
| Molecular Weight | 372.77 |